Ingredient intelligence

Retinol

Retinoid · Retinol · C20H30O

Retinol is a vitamin A alcohol that cells can convert to retinaldehyde and then retinoic acid, the form that binds nuclear retinoic acid receptors and changes gene transcription.

Molecular identity

Two-dimensional chemical structure of Retinol
Formula
C20H30O
Molecular weight
286.5 g/mol
PubChem CID
445354
ChEBI
CHEBI:17336
Open PubChem record →

Biological targets

  • Retinoic acid receptor alpha (RARA)

    high confidence

    activates · receptor

    Activated by the retinoic acid metabolite rather than retinol itself.

    UniProt P10276
  • Retinoic acid receptor gamma (RARG)

    high confidence

    activates · receptor

    UniProt P13631
  • Retinol dehydrogenase (RDH12)

    medium confidence

    targets · enzyme

    UniProt Q96NR8
  • Cellular retinol-binding protein 1 (RBP1)

    medium confidence

    targets · transporter

    UniProt P09455

Molecules & genes

Molecules

  • RetinolC20H30O · 286.5 g/mol
  • RetinaldehydeC20H28O · 284.4 g/mol
  • All-trans retinoic acidC20H28O2 · 300.4 g/mol

Genes / proteins

How could this ingredient interact with biology?

Biological network

Ingredient → molecule → target → gene/protein → pathway → process → studied outcome. Relationship strength is drawn from the curated confidence tier; nothing is added to make the chain look complete.

100%
RetinolRetinolRetinaldehydeAll-trans retinoic acidRetinoic acid receptor al…Retinoic acid receptor ga…Retinol dehydrogenase (RD…Cellular retinol-binding …RARARARGCOL1A1MMP1Retinoid metabolism and t…Nuclear receptor transcri…Extracellular matrix orga…Keratinocyte proliferationCollagen biosynthesisEpidermal cell turnoverStudied for photoaging-re…Studied for epidermal ren…Irritation and photosensi…

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IngredientMoleculeTargetGenePathwayProcessOutcome
Text alternative for this network
  • Retinol is molecule Retinolhigh confidence
  • Retinol is molecule Retinaldehydehigh confidence
  • Retinol is molecule All-trans retinoic acidhigh confidence
  • Retinol activates Retinoic acid receptor alpha (RARA)high confidence
  • Retinol activates Retinoic acid receptor gamma (RARG)high confidence
  • Retinol targets Retinol dehydrogenase (RDH12)medium confidence
  • Retinol targets Cellular retinol-binding protein 1 (RBP1)medium confidence
  • Retinoic acid receptor alpha (RARA) encoded by RARAhigh confidence
  • Retinoic acid receptor gamma (RARG) encoded by RARGhigh confidence
  • RARA participates in Retinoid metabolism and transporthigh confidence
  • RARG participates in Retinoid metabolism and transporthigh confidence
  • COL1A1 participates in Retinoid metabolism and transportmedium confidence
  • MMP1 participates in Retinoid metabolism and transportmedium confidence
  • RARA participates in Nuclear receptor transcription pathwayhigh confidence
  • RARG participates in Nuclear receptor transcription pathwayhigh confidence
  • COL1A1 participates in Nuclear receptor transcription pathwaymedium confidence
  • MMP1 participates in Nuclear receptor transcription pathwaymedium confidence
  • RARA participates in Extracellular matrix organisationmedium confidence
  • RARG participates in Extracellular matrix organisationmedium confidence
  • COL1A1 participates in Extracellular matrix organisationmedium confidence
  • MMP1 participates in Extracellular matrix organisationmedium confidence
  • Retinoid metabolism and transport associated with Keratinocyte proliferationhigh confidence
  • Nuclear receptor transcription pathway associated with Keratinocyte proliferationhigh confidence
  • Extracellular matrix organisation associated with Keratinocyte proliferationmedium confidence
  • Retinoid metabolism and transport associated with Collagen biosynthesismedium confidence
  • Nuclear receptor transcription pathway associated with Collagen biosynthesismedium confidence
  • Extracellular matrix organisation associated with Collagen biosynthesismedium confidence
  • Retinoid metabolism and transport associated with Epidermal cell turnoverhigh confidence
  • Nuclear receptor transcription pathway associated with Epidermal cell turnoverhigh confidence
  • Extracellular matrix organisation associated with Epidermal cell turnovermedium confidence
  • Keratinocyte proliferation studied in Studied for photoaging-related skin texture and wrinklingmedium confidence
  • Collagen biosynthesis studied in Studied for photoaging-related skin texture and wrinklingmedium confidence
  • Epidermal cell turnover studied in Studied for photoaging-related skin texture and wrinklingmedium confidence
  • Keratinocyte proliferation studied in Studied for epidermal renewalmedium confidence
  • Collagen biosynthesis studied in Studied for epidermal renewalmedium confidence
  • Epidermal cell turnover studied in Studied for epidermal renewalmedium confidence
  • Keratinocyte proliferation studied in Irritation and photosensitivity are commonly reported in studiesmedium confidence
  • Collagen biosynthesis studied in Irritation and photosensitivity are commonly reported in studiesmedium confidence
  • Epidermal cell turnover studied in Irritation and photosensitivity are commonly reported in studiesmedium confidence

Biological pathways

Retinoid metabolism and transport

high confidence

Conversion and carrier-protein handling of retinol and its metabolites.

Reactome R-HSA-975634

Nuclear receptor transcription pathway

high confidence

RAR/RXR heterodimers bind retinoic acid response elements and alter transcription.

Reactome R-HSA-383280

Extracellular matrix organisation

medium confidence

Collagen and matrix-metalloproteinase gene expression changes reported in retinoid-treated skin.

Reactome R-HSA-1474244

Evidence engine

Strong

Multiple independent human studies point in the same direction.

Skinceptor Evidence Index

77

experimental · of 100

This index is a research-navigation aid describing how much evidence exists and how it was produced. It is not a medical safety score, an efficacy guarantee, or a clinical recommendation.

Study composition

  • Human1
  • Randomised controlled trial2
  • Review1
Total studies
4
Human studies
3
Largest sample
44
Range
2000–2019

Index breakdown

  • Study design quality74% × 28%

    Mean design weight across curated studies (meta-analysis 1.0, RCT 0.9, other human 0.7, review 0.45, animal 0.35, in-vitro 0.25).

  • Human evidence share100% × 22%

    Proportion of curated evidence measured in people rather than cells or animals.

  • Evidence volume73% × 14%

    Log-scaled count of curated studies, so volume alone cannot dominate the score.

  • Largest sample size55% × 12%

    Log-scaled largest reported sample size across curated human studies.

  • Replication100% × 12%

    Independent human studies, capped at three; one study is never treated as replicated.

  • Recency65% × 7%

    Linear decay over a twenty-year window from the most recent curated publication.

  • Source traceability25% × 5%

    Share of curated studies with a verified PMID or DOI in this dataset.

How is this determined? →

Insufficient comparable evidence for quantitative synthesis.

Research timeline

How the evidence accumulated

  1. 2000

    Retinoid-induced procollagen synthesis and matrix metalloproteinase suppression in human skin in vivo

    Humann = 22 · Journal of Clinical Investigation

  2. 2007

    Retinol improves the appearance of naturally aged skin

    Randomised controlled trialn = 36 · Archives of Dermatology

  3. 2015

    Retinoic acid receptor expression and retinoid signalling in human skin

    Reviewsample size unavailable · Journal of Investigative Dermatology (review)

  4. 2019

    Prospective randomized double-blind assessment of topical bakuchiol and retinol for facial photoaging

    Randomised controlled trialn = 44 · British Journal of Dermatology

Ingredient fingerprint

21 nodes · 41 relationships · seed "retinol"

The fingerprint is a deterministic visual signature: ridge amplitude comes from the number of entities in each tier, node placement from identifier hashes, and opacity from confidence. Two ingredients can never produce the same figure unless their networks are identical.

Open in Biology as Art →

Research

4 curated studies

Randomised controlled trialBritish Journal of Dermatology · 2019n = 44

Prospective randomized double-blind assessment of topical bakuchiol and retinol for facial photoaging

Reported comparable improvement in wrinkle and pigmentation scores between bakuchiol and retinol, with less scaling and stinging reported for bakuchiol.

LimitationsSingle centre, 12 weeks, no vehicle arm, so both may reflect regression to the mean.

PMID 29752709Bakuchiol · Retinol
ReviewJournal of Investigative Dermatology (review) · 2015

Retinoic acid receptor expression and retinoid signalling in human skin

Summarises RAR/RXR heterodimer signalling as the transcriptional mechanism of retinoid action in epidermis and dermis.

LimitationsNarrative review; mechanistic focus without effect-size synthesis.

Identifier not curated — search Europe PMCRetinol · All-trans retinoic acid · Retinaldehyde
Randomised controlled trialArchives of Dermatology · 2007n = 36

Retinol improves the appearance of naturally aged skin

Reported improvement in fine wrinkling with topical retinol versus vehicle in older adults.

LimitationsSmall sample; older cohort limits generalisation; identifier not verified during curation.

HumanJournal of Clinical Investigation · 2000n = 22

Retinoid-induced procollagen synthesis and matrix metalloproteinase suppression in human skin in vivo

Reported increased procollagen I expression and reduced MMP-1 in biopsied retinoid-treated skin.

LimitationsBiopsy-based surrogate endpoints; identifier not verified during curation.

Identifier not curated — search Europe PMCAll-trans retinoic acid · Retinol

Community evidence

Submitted by readers

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Reader submissions appear here only after review. They are not part of the curated dataset and do not affect the Skinceptor Evidence Index.

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Sources